| GENIPOSIDIC-ACID | ED50=>800 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| DEACETYLASPERULOSIDIC-ACID | ED50=>600 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| MONOTROPEIN | ED50=>500 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| CATALPOSIDE | ED50=>300 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| DEOXYGENIPOSIDE | ED50=>1,200 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| DEOXYLOGANIN | ED50=800 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| LOGANIN | ED50=540 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| DEACETYLASPERULOSIDIC-ACID-METHYL-ESTER | ED50=530 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| AUCUBIN | ED50=390 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| CATALPOL | ED50=340 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| GENIPOSIDE | ED50=300 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| PAEDEROSIDE | ED50=300 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| ASPERULOSIDE | ED50=240 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| PLUMIERIDE | ED50=120 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| VERBENALIN | ED50=110 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| GARDENOSIDE | ED50=1,200 mg/kg | Wagner & Wolff, eds. 1977. New Natural Products (RS164. I56. 176) |
| ELATERIN | 3-6 mg/man | * |
| ALOE-EMODIN | -- | Merck 11th Edition |
| LIGNANS | -- | * |
| FRANGULIN | -- | Merck 11th Edition |
| PRUNUSIDE | -- | * |
| ARECOLINE | -- | Merck 11th Edition |
| CHRYSOPHANOL | -- | * |
| SENNIDIN | -- | * |
| OXYSPARTEINE | -- | * |
| GLUCO-FRANGULIN | -- | Merck 11th Edition |
| SORBITOL | -- | * |
| CASANTHRANOL | -- | Merck 11th Edition |
| PHYSCION | -- | * |
| 4'-DEMETHYLPODOPHYLLUM | -- | Jeffery B. Harborne and H. Baxter, eds. 1983. Phytochemical Dictionary. A Handbook of Bioactive Compounds from Plants. Taylor & Frost, London. 791 pp. |
| KOSAMIN | -- | * |
| SPARTEINE | -- | * |
| EMODIN | -- | Merck 11th Edition |
| PODOPHYLLOTOXIN | -- | Jeffery B. Harborne and H. Baxter, eds. 1983. Phytochemical Dictionary. A Handbook of Bioactive Compounds from Plants. Taylor & Frost, London. 791 pp. |
| ANAGYRINE | -- | * |
| LUPININE | -- | * |
| CHRYSAZIN | -- | Jeffery B. Harborne and H. Baxter, eds. 1983. Phytochemical Dictionary. A Handbook of Bioactive Compounds from Plants. Taylor & Frost, London. 791 pp. |
| RHEIN | -- | * |
| MYCORINEMATARESINOL-MONOGLUCOSIDE | -- | * |
| SENNOSIDE | -- | * |
| BETA-GUTTIFERIN | -- | * |
| IRIDIN | -- | * |
| CASCAROSIDE-A | -- | Jeffery B. Harborne and H. Baxter, eds. 1983. Phytochemical Dictionary. A Handbook of Bioactive Compounds from Plants. Taylor & Frost, London. 791 pp. |